BX912 is a potent and specific PDK1 inhibitor with IC50 of 12 nM, 9- and 105- fold greater selectivity for PKD1 than PKA and PKC, respectively. In comparison to GSK3¦Â, selectivity for PDK1 is 600-fold.

June 21, 2017

prudect name : BX912 is a potent and specific PDK1 inhibitor with IC50 of 12 nM, 9- and 105- fold greater selectivity for PKD1 than PKA and PKC, respectively. In comparison to GSK3¦Â, selectivity for PDK1 is 600-fold.
BX-912 BX912;BX 912

Synonyms: CAS NO: 702674-56-4Molecular Formula: C₂₀H₂₃BrN₈OMolecular Weight: 471.36Purity: 98% minSolubility: In DMSOStorage: -20°C

EPZ-015666 References PubMed ID：:http://www.ncbi.nlm.nih.gov/pubmed/18503759