GSK-LSD1 2HCl is an irreversible, and selective LSD1 inhibitor with IC50 of 16 nM, > 1000 fold selective over other closely related FAD utilizing enzymes (i.e. LSD2, MAO-A, MAO-B).

June 21, 2017

prudect name : GSK-LSD1 2HCl is an irreversible, and selective LSD1 inhibitor with IC50 of 16 nM, > 1000 fold selective over other closely related FAD utilizing enzymes (i.e. LSD2, MAO-A, MAO-B).
GSK-LSD1 (LSD1 inhibitor)

Synonyms: CAS NO: 1431368-48-7Molecular Formula: C₁₄H₂₀N₂Molecular Weight: 216.32Purity: 98% minSolubility: DMSOStorage: -20¡æ

Prexasertib References PubMed ID：:http://www.ncbi.nlm.nih.gov/pubmed/18518824