ENMD-2076 tartrate has selective activity against Aurora A and Flt3 with IC50 of 14 nM and 1.86 nM, 25-fold selective for Aurora A than over Aurora B and less potent to VEGFR2/KDR and VEGFR3, FGFR1 and FGFR2 and PDGFR¦Á.

June 21, 2017

prudect name : ENMD-2076 tartrate has selective activity against Aurora A and Flt3 with IC50 of 14 nM and 1.86 nM, 25-fold selective for Aurora A than over Aurora B and less potent to VEGFR2/KDR and VEGFR3, FGFR1 and FGFR2 and PDGFR¦Á.
ENMD-2076 Tartrate

Synonyms: CAS NO: 1291074-87-7Molecular Formula: C₂₁H₂₅N₇.x(C₄H₆O₆)Molecular Weight: 1291074-87-7Purity: 98% minSolubility: in DMSOStorage: -20oC

BGJ-398 References PubMed ID：:http://www.ncbi.nlm.nih.gov/pubmed/18513435