Dorsomorphin is a potent, reversible, selective AMPK inhibitor with Ki of 109 nM in cell-free assays, exhibiting no significant inhibition of several structurally related kinases including ZAPK, SYK, PKC¦È, PKA, and JAK3. Also inhibits type I BMP receptor activity.

June 21, 2017

prudect name : Dorsomorphin is a potent, reversible, selective AMPK inhibitor with Ki of 109 nM in cell-free assays, exhibiting no significant inhibition of several structurally related kinases including ZAPK, SYK, PKC¦È, PKA, and JAK3. Also inhibits type I BMP receptor activity.
Dorsomorphin

Synonyms: BML-275CAS NO: 866405-64-3Molecular Formula: C₂₄H₂₅N₅OMolecular Weight: 399.49Purity: 98% minSolubility: In DMSOStorage: −20°C 2 years

1,1-Dimethylbiguanide hydrochloride References PubMed ID：:http://www.ncbi.nlm.nih.gov/pubmed/18509765