Biological Activity Potent, selective and competitive P2X7 receptor antagonist (IC50 values are 18 and 40 nM for rat and human receptors respectively). Displays selectivity over a variety of P2X and P2Y receptors up to a concentration of 100 ¦ÌM. Reduces nociception in animal models of persistent neuropathic and inflammatory pain.

June 21, 2017

prudect name : Biological Activity
Potent, selective and competitive P2X7 receptor antagonist (IC50 values are 18 and 40 nM for rat and human receptors respectively). Displays selectivity over a variety of P2X and P2Y receptors up to a concentration of 100 ¦ÌM. Reduces nociception in animal models of persistent neuropathic and inflammatory pain.
A-740003

Synonyms: CAS NO: 861393-28-4Molecular Formula: C₂₆H₃₀N₆O₃Molecular Weight: 474.55Purity: 98% minSolubility: In DMSOStorage: -20°C

1373423-53-0 References PubMed ID：:http://www.ncbi.nlm.nih.gov/pubmed/18497534